Author(s): Mule Asmita, Kote Rupali Balasaheb, Jadhav Ravindra S, Khemnar Ashwini, Jinat Maniyar, Khetmalis Aditya, Monika Magar, Nikita Borse

Email(s): rupalikote236@gmail.com

DOI: 10.52711/2321-5836.2026.00014   

Address: Mule Asmita*, Kote Rupali Balasaheb, Jadhav Ravindra S, Khemnar Ashwini, Jinat Maniyar, Khetmalis Aditya, Monika Magar, Nikita Borse
Department of Pharmaceutics, Pravara Rural Education Society's Institute of Pharmacy, Loni.
*Corresponding Author

Published In:   Volume - 18,      Issue - 1,     Year - 2026


ABSTRACT:
Ocular drug delivery remains one of the major challenges in pharmaceutical research due to the complex anatomy and physiology of the eye. The eye, being a delicate and highly protected organ responsible for vision, presents various barriers that hinder effective drug absorption. The purpose of ocular drug delivery systems is to achieve therapeutic concentrations of drugs at the target site while minimizing systemic exposure and side effects. This review discusses the anatomy of the eye relevant to drug delivery, various routes of ocular administration, physiological barriers, dosage forms, and recent advancements in ocular delivery technologies. The advantages, limitations, and marketed products for different ocular dosage forms are also reviewed. The review further highlights recent innovations such as in-situ gels, nanoparticles, and implants, which offer controlled and sustained release profiles for improved therapeutic efficacy.


Cite this article:
Mule Asmita, Kote Rupali Balasaheb, Jadhav Ravindra S, Khemnar Ashwini, Jinat Maniyar, Khetmalis Aditya, Monika Magar, Nikita Borse. A Review on Ocular Drug Delivery System. Research Journal of Pharmacology and Pharmacodynamics. 2026;18(1):107-0. doi: 10.52711/2321-5836.2026.00014

Cite(Electronic):
Mule Asmita, Kote Rupali Balasaheb, Jadhav Ravindra S, Khemnar Ashwini, Jinat Maniyar, Khetmalis Aditya, Monika Magar, Nikita Borse. A Review on Ocular Drug Delivery System. Research Journal of Pharmacology and Pharmacodynamics. 2026;18(1):107-0. doi: 10.52711/2321-5836.2026.00014   Available on: https://www.rjppd.org/AbstractView.aspx?PID=2026-18-1-14


REFERENCES:
1.    Patel A, Cholkar K, Agrahari V, Mitra AK. Ocular drug delivery systems: An overview. World J Pharmacol. 2013; 2(2): 47–64.
2.    Singh M, Tyagi S, Verma R. Recent advances in ocular drug delivery systems. Res J Pharmacodyn Pharmacol. 2020; 12(1):33–42.
3.    Nanjwade BK, et al. Development and evaluation of in-situ gelling systems for ocular drug delivery. Res J Pharmacodyn Pharmacol. 2019; 11(3): 127–134.
4.    Kumar S, et al. Nanotechnology in ophthalmic drug delivery. Res J Pharmacodyn Pharmacol. 2021; 13(2): 55–63.
5.    Jain R, et al. Ocular barriers and strategies to overcome them. Int J Pharm Sci Res. 2018; 9(4): 1345–1353.
6.    Shinde GS, Rao PS, Jadhav RS, Kolhe P, Athare D. A review on chromatography and advancement in paper chromatography technique. Asian Journal of Pharmaceutical Analysis. 2021; 11(1): 45-8
7.    Chauhan A, Radke CJ. Controlled release of drugs from ophthalmic delivery systems. Adv Drug Deliv Rev. 2012; 64(6): 666–685.
8.    Shinde, G. S., Jadhav, R., Vikhe, D., and Kote, R. B. Development and evaluation of herbal fast disintegrating tablet of Achyranthes aspera linn root extract. Asian Journal of Pharmacy and Technology, 2024: 14(2): 119-122.
9.    Shinde, G. S, Jadhav R S, Tambe V B, Kote R B .RP-HPLC Method Development and Validation of Lamivudine, Zidovudine and Nevirapine in Bulk and Dosage form using UV Detector." Research Journal of Pharmacy and Technology. 2024; 17(10): 5011-5015
10.    Suresh PK, Barsa G, Sah AK, Daharwal SJ. Ocular implants as drug delivery device in ophthalmic therapeutics: An overview. Res J Pharm Technol. 2014; 7(6): 687–693.
11.    Shinde GS, Jadhav RS, Kote RB, Kadam AJ, Bankar AA. Bioanalytical Method Development and Validation of UV Spectrophotometric Method for Estimation of Metformin Hydrochloride in Urine Sample. Asian J Res Chem. 2024; 17(2): 93–6. doi: 10.52711/0974-4150.2024.00019
12.    Karthikeyan D, Vijaikumar S, Pandey VP, Nandha Kumar J, Sengottuvelu S, Shivakumar T. Preparation and evaluation of ocular inserts for controlled delivery of Ciprofloxacin hydrochloride. Res J Pharm Technol. 2008; 1(1): 37–41.
13.    Nautiyal D, Singh V, Ali S. Formulation and evaluation of sustained release of Ofloxacin ocular inserts. Res J Pharm Technol. 2012; 5(12): 1533–1538.
14.    Karthikeyan D, Sonkar S, Pandey VP, Nandha Kumar J, Sengottuvelu S, Bhowmick M, Shivakumar T. Development and characterization of modified ocular inserts with improved ocular compatibility. Res J Pharm Technol. 2008; 1(2): 93–99.
15.    Godge RK, Shinde GS, Joshi S. Simultaneous Estimation and Validation of Dapagliflozin and Saxagliptin in Bulk Drug and Dosage Form by RP-HPLC. Research Journal of Science and Technology. 2019; 11(1):59-63
16.    Gupta SK, Singhvi IL. In-situ gelling system and other possible innovative approach for ocular disease: A review. Res J Pharm Technol. 2011; 4(6): 825–829.
17.    Shinde V, Amsa P, Tamizharasi S, Karthikeyan D, Shivakumar T, Kale A. Formulation and characterization of Eudragit RS 100 nanosuspension for ocular delivery of indomethacin. Res J Pharm Technol. 2010;3(3):779–784.
18.    Nayak S, Jadhav M, Bhaskar V. Recent advances in ocular drug delivery system. Res J Pharm Technol. 2016; 9(7): 789–795.
19.    Shinde G, Godage RK, Jadhav RS, Manoj B, Aniket B. A Review on Advances in UV Spectroscopy. Research Journal of Science and Technology. 2020; 12(1): 47-51.
20.    Nair RV, Nair SC, Anoop KR. Current trends in ocular drug systems and its applications. Res J Pharm Technol. 2015; 8(5): 589–595.
21.    Pawar P, Yadav A, Gharge V. Ocular drug delivery and novel formulation: A review. Asian J Pharm Technol. 2018; 8(4): 218–224

Recomonded Articles:

Author(s): Purnendu Panda, Indu.S, Banamali Das, G.C. Bhuyan, M.M. Rao

DOI: 10.52711/2321-5836.2022.00047         Access: Open Access Read More

Author(s): Aswani P. S., Kshirod Kumar Ratha, Dighe Dattatray Pandurang, M. M. Rao, Remya Vijayan

DOI: 10.5958/2321-5836.2018.00008.3         Access: Open Access Read More

Author(s): Purnendu Panda, Banamali Das, DS Sahu, SK Meher, Das, GC Nanda.

DOI: Not Available         Access: Open Access Read More

Author(s): Shameer Pasha, Mohamed Khaleel, Sukhen Som.

DOI: Not Available         Access: Open Access Read More

Author(s): Sachin Aglawe, Amol Gayke, Kavita Sharma, Sonali Jadhav, Sanjivani Gore, Bhagyashri Pandit, Sonali Valate, Mayuri Wagh

DOI: 10.5958/2321-5836.2020.00003.8         Access: Open Access Read More

Author(s): Ganesh G. Dhakad, Megha S. Nannaware, Gauri V. Wagh, Abhijit V. Shrirao, N.I. Kochar, A.V. Chandewar

DOI: 10.52711/2321-5836.2023.00012         Access: Open Access Read More

Author(s): S. D. Kadam, S. A. Chavhan, S. A. Shinde, P. N. Sapkal

DOI: 10.5958/2321-5836.2018.00032.0         Access: Open Access Read More

Author(s): Sanjib Kumar Das, Anuradha Das, Banamali Das, Purnendu Panda, G. C. Bhuyan, Bipin Bihari Khuntia

DOI: 10.5958/2321-5836.2017.00036.2         Access: Open Access Read More

Author(s): Jeena S, Venkateswaramurthy N, Sambathkumar R

DOI: 10.5958/2321-5836.2020.00004.X         Access: Open Access Read More

Author(s): Pallavi B. Jire, Mayuri V. Khairnar, Mayuri V. Mali, Sulbha G. Patil

DOI: 10.52711/2321-5836.2023.00024         Access: Open Access Read More

Author(s): U. S. Jijith , C. R. Sudhakaran Nair, K. Pramod

DOI: 10.5958/2321-5836.2016.00001.X         Access: Open Access Read More

Author(s): S. Anandkumar, Jessly Chacko, Theertha C. K, M. Usha

DOI: 10.5958/2321-5836.2020.00001.4         Access: Open Access Read More

Author(s): Rohit J. Bhor, Harshala Damdhar, Geeta Kokate, Maduri Salve, Swati Andhale

DOI: 10.5958/2321-5836.2016.00025.2         Access: Open Access Read More

Author(s): K. Sanjeev Kumar, V Vijay Kumar, AG Prasanthi, LK Kanthal, P Bhoja Raju, K Satyavathi .

DOI: Not Available         Access: Open Access Read More

Author(s): Divyashree Kantilal Patil, Divyani Rajendra Patil, Sunila A. Pati

DOI: 10.52711/2321-5836.2023.00015         Access: Open Access Read More

Author(s): Suneel Kumar A, Venkatarathanamma. V, Naga Saibabu V, Nageswara Rao Tentu, Pavan Kumar Kota, K. Suneel Kumar, A. Vijayalakshmi

DOI: 10.5958/2321-5836.2017.00009.X         Access: Open Access Read More

Author(s): Neeraj Vyawahare, Virendra Kagathara, Rohini Pujari, Manoj Patil, Imtiyaz Ansari and Amol Bhandare.

DOI: Not Available         Access: Open Access Read More

Research Journal of Pharmacology and Pharmacodynamics (RJPPD) is an international, peer-reviewed journal....... Read more >>>

RNI: Not Available                     
DOI: 10.5958 2321-5836 

Journal Policies & Information




Recent Articles




Tags